IV (n = 5) | SC (n = 5) | |
---|---|---|
Dose (mg/kg) | 0.05 | 1.00 |
t1/2 (h) | 3.67 ± 0.40 | 3.55 ± 0.51 |
C0 or Cmax (ng/mL) | 822.08 ± 227.19 | 669.64 ± 186.57 |
Tmax (h)* | – | 3.00 (2.00–6.00) |
AUCall (ng·h/mL) | 3429.30 ± 875.27 | 9166.62 ± 2465.16 |
AUCinf (ng·h/mL) | 3505.33 ± 815.04 | 9223.30 ± 2417.73 |
CL or CL/F (mL/min/kg) | 0.25 ± 0.06 | 1.92 ± 0.52 |
Vss (mL/kg) | 73.12 ± 20.68 | – |
Bioavailability | – | 13.16% |