Formulation code | In vitro studies | Ex vivo studies | ||||
---|---|---|---|---|---|---|
Slope | Permeability coefficient (cm/h) | Flux (μg/cm2/h) | Slope | Permeability coefficient (cm/h) | Flux (μg/cm2/h) | |
A1 | 0.554 | 0.0122 | 176.43 | 0.435 | 0.0095 | 138.53 |
A2 | 0.536 | 0.0118 | 170.70 | 0.39 | 0.0085 | 124.20 |
A3 | 0.536 | 0.0118 | 170.70 | 0.349 | 0.0076 | 111.14 |
A4 | 0.499 | 0.0109 | 158.91 | 0.316 | 0.0069 | 100.63 |
B1 | 0.557 | 0.0122 | 177.38 | 0.405 | 0.0089 | 128.98 |
B2 | 0.524 | 0.0115 | 166.87 | 0.377 | 0.0083 | 120.06 |
B3 | 0.476 | 0.0104 | 151.59 | 0.345 | 0.0075 | 109.87 |
B4 | 0.494 | 0.0108 | 157.32 | 0.321 | 0.0070 | 102.22 |
C1 | 0.549 | 0.0120 | 174.84 | 0.518 | 0.0114 | 164.96 |
C2 | 0.565 | 0.0124 | 179.93 | 0.493 | 0.0108 | 157.00 |
C3 | 0.524 | 0.0115 | 166.87 | 0.485 | 0.0106 | 154.45 |
C4 | 0.521 | 0.0114 | 165.92 | 0.437 | 0.0096 | 139.17 |